Abstract
A palladium-catalyzed intramolecular amination of alkenes with retention of olefin functionalization was achieved under mild reaction conditions. In the presence of palladium catalyst, the tosyl-protected amine can directly couple with a double bond to provide versatile dihydropyrrole derivatives in moderate to excellent yields.
Original language | English |
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Pages (from-to) | 914-917 |
Number of pages | 4 |
Journal | Organic Letters |
Volume | 19 |
Issue number | 4 |
DOIs | |
State | Published - 17 Feb 2017 |
Externally published | Yes |