Copper(I) Iodide-Catalyzed (Het)arylation of Diethyl Malonate with (Het)aryl Bromides by Using 1,3-Benzoxazole as a Ligand

Yu Zeng, Hao Liang Zheng, Zhao Yang, Cheng Kou Liu, Zheng Fang, Kai Guo

科研成果: 期刊稿件文章同行评审

4 引用 (Scopus)

摘要

An efficient Ullmann-type coupling of aryl bromides with diethyl malonate in the presence of copper(I) iodide and 1,3-benzoxazole is presented. This method has a broad substrate scope (heterocyclic and phenyl bromides) and good functional-group tolerance (OMe, Me, Ac, CN, NO 2, F, and Cl). Moreover, less time is needed to reach full conversion (3-9 hours).

源语言英语
文章编号st-2017-w0499-l
页(从-至)79-84
页数6
期刊Synlett
29
1
DOI
出版状态已出版 - 3 1月 2018

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