Design, synthesis and biological evaluation of Sunitinib analogues to improve aqueous solubility

Ke Tao Chen, Zheng Fang, Zhao Yang, Kai Guo

科研成果: 书/报告/会议事项章节会议稿件同行评审

4 引用 (Scopus)

摘要

In order to improve aqueous solubility of Sunitinib, based on the structure-activity relationship, four analogues were designed and synthesized. The obtained structures were identified by 1H NMR, MS and elemental analysis. In vitro evaluation of antitumor bioactivity was performed by MTT method. All of synthesized compounds showed antitumor activities, especially, compounds A1, which were better than or equal to the antitumor activity of positive control.

源语言英语
主期刊名Bio-Medical Materials and Engineering
350-353
页数4
DOI
出版状态已出版 - 2013
活动2013 International Conference on Bio-Medical Materials and Engineering, ICBME 2013 - Hong Kong, 中国
期限: 26 3月 201327 3月 2013

出版系列

姓名Advanced Materials Research
749
ISSN(印刷版)1022-6680

会议

会议2013 International Conference on Bio-Medical Materials and Engineering, ICBME 2013
国家/地区中国
Hong Kong
时期26/03/1327/03/13

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