Iron-catalyzed [4 + 2] annulation of amidines with α,β-unsaturated ketoxime acetates toward 2,4,6-trisubstituted pyrimidines

Qinghuan Wu, Luchao Li, Binyan Xu, Jie Sun, Dong Ji, Yuguang Li, Lei Shen, Zheng Fang, Jindian Duan, Beining Chen, Kai Guo

科研成果: 期刊稿件文章同行评审

4 引用 (Scopus)

摘要

An iron-catalyzed [4 ​+ ​2] annulation of amidines with α,β-unsaturated ketoxime acetates is described. This strategy employs amidines as CN units and provides a new protocol for the construction of 2,4,6-trisubstituted pyrimidines under batch and continuous flow conditions in moderate to good yields, exhibiting good functional group tolerance, scalability and operational simplicity.

源语言英语
页(从-至)150-153
页数4
期刊Green Synthesis and Catalysis
4
2
DOI
出版状态已出版 - 5月 2023

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