Synthesis of Alkylsulfonyl-Substituted Indolo[2,1-a]Isoquinolines via Photoredox-Catalyzed Radical-Cascade Addition/Sulfonylation/Cyclization with DABCO ⋅ (SO2)2 and Thianthrenium Salts

Xin Yuan, Jie Liu, Long Zhou Qin, Xiu Duan, Jian Wang, Meng Yu Wu, Jiang Kai Qiu, Kai Guo

科研成果: 期刊稿件文章同行评审

13 引用 (Scopus)

摘要

A direct, visible-light-mediated, radical-cascade addition/sulfonylation/cyclization reaction with DABCO ⋅ (SO2)2 and thianthrenium salts is reported herein. This protocol provides operationally-convenient access to various sulfonated functionalized indole [2,1-a] isoquinolines under mild conditions. This transformation features high functional-group tolerance, operational ease, and broad substrate scope. Preliminary studies reveal that the method undergoes a radical pathway. (Figure presented.).

源语言英语
页(从-至)555-567
页数13
期刊Advanced Synthesis and Catalysis
365
4
DOI
出版状态已出版 - 21 2月 2023

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