Bisintercalator-containing dinuclear iron(III) complex: An efficient artificial nuclease

Xiaoqiang Chen, Jiangli Fan, Xiaojun Peng, Jingyun Wang, Shiguo Sun, Rong Zhang, Tong Wu, Fei Zhang, Jianfeng Liu, Fen Wang, Saijian Ma

科研成果: 期刊稿件文章同行评审

14 引用 (Scopus)

摘要

Two acridine groups were successfully introduced into di-iron(III) complex. DNA cleavage experiments indicated that complex conjugating bisacridine groups can enhance 300-fold for the cleavage efficiency compared with complex lacking of acridine conjugation. Further ligation assay of DNA segments provided the evidence for hydrolytic mechanism of DNA cleavage.

源语言英语
页(从-至)4139-4142
页数4
期刊Bioorganic and Medicinal Chemistry Letters
19
15
DOI
出版状态已出版 - 1 8月 2009
已对外发布

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