TY - JOUR
T1 - Cu-catalyzed direct C-H bond functionalization
T2 - A regioselective protocol to 5-aryl thiazolo[3,2-b]-1,2,4-triazoles
AU - Xie, Zengyang
AU - Zhu, Xiaojun
AU - Guan, Yangfan
AU - Zhu, Dunru
AU - Hu, Hongwen
AU - Lin, Chen
AU - Pan, Yi
AU - Jiang, Juli
AU - Wang, Leyong
PY - 2013/2/28
Y1 - 2013/2/28
N2 - An efficient, regioselective C-5 arylation of thiazolo[3,2-b]-1,2,4- triazoles catalyzed by a simple copper catalyst was developed. This arylation proceeded smoothly and tolerated a variety of functional groups (44 examples). A wide range of functionalized thiazolo[3,2-b]-1,2,4-triazole derivatives were obtained in high yields (up to 99% yield). Possible catalytic cycles of the arylation were also discussed.
AB - An efficient, regioselective C-5 arylation of thiazolo[3,2-b]-1,2,4- triazoles catalyzed by a simple copper catalyst was developed. This arylation proceeded smoothly and tolerated a variety of functional groups (44 examples). A wide range of functionalized thiazolo[3,2-b]-1,2,4-triazole derivatives were obtained in high yields (up to 99% yield). Possible catalytic cycles of the arylation were also discussed.
UR - http://www.scopus.com/inward/record.url?scp=84875860155&partnerID=8YFLogxK
U2 - 10.1039/c2ob27326h
DO - 10.1039/c2ob27326h
M3 - 文章
C2 - 23328869
AN - SCOPUS:84875860155
SN - 1477-0520
VL - 11
SP - 1390
EP - 1398
JO - Organic and Biomolecular Chemistry
JF - Organic and Biomolecular Chemistry
IS - 8
ER -