Synthesis and bioactivity of novel 2-(1,2-benzisothiazol-3-yloxy)-N-(1-aryl-3-cyanopyrazol-5-yl) acetamides

Peng Yu; Xi Li; Xiao Zhang; Yanhua Xu

doi:10.24820/ARK.5550190.P011.091

Synthesis and bioactivity of novel 2-(1,2-benzisothiazol-3-yloxy)-N-(1-aryl-3-cyanopyrazol-5-yl) acetamides

Peng Yu, Xi Li, Xiao Zhang, Yanhua Xu

环境科学与工程学院

Nanjing Tech University

科研成果: 期刊稿件 › 文章 › 同行评审

摘要

Nine novel types of 2-(1,2-benzisothiazol-3-yloxy)-N-(1-aryl-3-cyanopyrazol-5-yl)-acetamides were synthesized, and their inhibition effects on selected bacteria (heterotrophic bacteria) and algae (marine chlorella) were evaluated. Results showed that 2-(1,2-benzisothiazol-3-yloxy)-N-(3-cyano-1-(2,4-dimethylphenyl)pyrazol-5-yl) acetamide achieved the highest yield of 81% with good bioactivity against heterotrophic bacteria and marine chlorella.

源语言	英语
页（从-至）	397-405
页数	9
期刊	Arkivoc
卷	2019
期	6
DOI	https://doi.org/10.24820/ARK.5550190.P011.091
出版状态	已出版 - 1月 2020

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10.24820/ARK.5550190.P011.091

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title = "Synthesis and bioactivity of novel 2-(1,2-benzisothiazol-3-yloxy)-N-(1-aryl-3-cyanopyrazol-5-yl) acetamides",

abstract = "Nine novel types of 2-(1,2-benzisothiazol-3-yloxy)-N-(1-aryl-3-cyanopyrazol-5-yl)-acetamides were synthesized, and their inhibition effects on selected bacteria (heterotrophic bacteria) and algae (marine chlorella) were evaluated. Results showed that 2-(1,2-benzisothiazol-3-yloxy)-N-(3-cyano-1-(2,4-dimethylphenyl)pyrazol-5-yl) acetamide achieved the highest yield of 81% with good bioactivity against heterotrophic bacteria and marine chlorella.",

keywords = "Bioactivity, Isothiazolinone, N-Aryl pyrazole, Synthesis",

author = "Peng Yu and Xi Li and Xiao Zhang and Yanhua Xu",

note = "Publisher Copyright: {\textcopyright} AUTHOR (S).",

year = "2020",

month = jan,

doi = "10.24820/ARK.5550190.P011.091",

language = "英语",

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TY - JOUR

T1 - Synthesis and bioactivity of novel 2-(1,2-benzisothiazol-3-yloxy)-N-(1-aryl-3-cyanopyrazol-5-yl) acetamides

AU - Yu, Peng

AU - Li, Xi

AU - Zhang, Xiao

AU - Xu, Yanhua

N1 - Publisher Copyright: © AUTHOR (S).

PY - 2020/1

Y1 - 2020/1

N2 - Nine novel types of 2-(1,2-benzisothiazol-3-yloxy)-N-(1-aryl-3-cyanopyrazol-5-yl)-acetamides were synthesized, and their inhibition effects on selected bacteria (heterotrophic bacteria) and algae (marine chlorella) were evaluated. Results showed that 2-(1,2-benzisothiazol-3-yloxy)-N-(3-cyano-1-(2,4-dimethylphenyl)pyrazol-5-yl) acetamide achieved the highest yield of 81% with good bioactivity against heterotrophic bacteria and marine chlorella.

AB - Nine novel types of 2-(1,2-benzisothiazol-3-yloxy)-N-(1-aryl-3-cyanopyrazol-5-yl)-acetamides were synthesized, and their inhibition effects on selected bacteria (heterotrophic bacteria) and algae (marine chlorella) were evaluated. Results showed that 2-(1,2-benzisothiazol-3-yloxy)-N-(3-cyano-1-(2,4-dimethylphenyl)pyrazol-5-yl) acetamide achieved the highest yield of 81% with good bioactivity against heterotrophic bacteria and marine chlorella.

KW - Bioactivity

KW - Isothiazolinone

KW - N-Aryl pyrazole

KW - Synthesis

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DO - 10.24820/ARK.5550190.P011.091

M3 - 文章

AN - SCOPUS:85093895349

SN - 1551-7004

VL - 2019

SP - 397

EP - 405

JO - Arkivoc

JF - Arkivoc

IS - 6

ER -

Synthesis and bioactivity of novel 2-(1,2-benzisothiazol-3-yloxy)-N-(1-aryl-3-cyanopyrazol-5-yl) acetamides

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